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GPCR & Ion Channel Stable Cell Lines

GenScript offers a large product portfolio covering GPCR and ion channel stable cell lines, as well as well other products made using these stable cell lines: Ready-to-UseTM Frozen Cells and Membrane Preparations. In addition, GenScript offers Custom Stable Cell Line Service upon your specifications.

GPCR Stable Cell Lines

Cat. No.
Cell Line
GPCR Family
Receptor
Price (USD)
Selected
CHO-K1/M1 Acetylcholine (muscarinic) M1 / CHRM1
$11,600.00
CHO-K1/M2/Gα15 Acetylcholine (muscarinic) M2 / CHRM2
$11,600.00
CHO-K1/M3 Acetylcholine (muscarinic) M3 / CHRM3
$11,600.00
CHO-K1/M4/Gα15 Acetylcholine (muscarinic) M4 / CHRM4
$11,600.00
CHO-K1/M5 Acetylcholine (muscarinic) M5 / CHRM5
$11,600.00
CHO-K1/ADORA1/Gα15 Adenosine ADORA1
$11,600.00
CHO-K1/ADORA2A/Gα15 Adenosine ADORA2A
$11,600.00
CHO-K1/ADORA2B/Gα15 Adenosine ADORA2B
$11,600.00
M00464
CHO-K1/ADORA3/Gqi5 Adenosine ADORA3
$11,600.00
Coming soon
CHO-K1/ADRA1A Adrenoceptors ADRA1A
$11,600.00
CHO-K1/ADRA1B Adrenoceptors ADRA1B
$11,600.00
CHO-K1/ADRA1D Adrenoceptors ADRA1D
$11,600.00
CHO-K1/ADRA2A/Gα15 Adrenoceptors ADRA2A
$11,600.00
M00454
CHO-K1/ADRA2B/Gqi5 Adrenoceptors ADRA2B
$11,600.00
Coming soon
CHO-K1/ADRA2C/Gα15 Adrenoceptors ADRA2C
$11,600.00
CHO-K1/ADRB1/Gα15 Adrenoceptors ADRB1
$11,600.00
CHO-K1/ADRB2/Gα15 Adrenoceptors ADRB2
$11,600.00
293/ADRB3/CRE-Luc Adrenoceptors ADRB3
$11,600.00
CHO-K1/C5a/Gα15 Anaphylotoxin C5a / C5AR1
$11,600.00
293T/AT1 Angiotensin AT1
$11,600.00
CHO-K1/AGTRL1/Gα15 Apelin AGTRL1
$11,600.00
CHO-K1/GPBAR1 Bile acid GPBAR1
$11,600.00
CHO-K1/BB1 Bombesin BB1 / NMBR
$11,600.00
CHO-K1/BB2 Bombesin BB2 / GRPR
$11,600.00
CHO-K1/BB3 Bombesin BB3 / BRS3
$11,600.00
CHO-K1/B2/Gα15 Bradykinin B2 / BDKRB2
$11,600.00
CHO-K1/CB1/Gα15 Cannabinoid CB1 / CNR1
$11,600.00
CHO-K1/CB2 Cannabinoid CB2 / CNR2
$11,600.00
CHO-K1/CMKLR1/Gα15 Chemoattractant ChemR23 / CMKLR1
$11,600.00
M00496
CHO-K1/CCR8/Gα15 Chemokine CCR8
$11,600.00
Coming soon
CHO-K1/CCKA/Gα15 Cholecystokinin CCKA
$11,600.00
CHO-K1/CCKB Cholecystokinin CCKB
$11,600.00
CHO-K1/D1 Dopamine D1 / DRD1
$11,600.00
CHO-K1/D2/Gα15 Dopamine D2 / DRD2
$11,600.00
CHO-K1/D2S/Gα15 Dopamine D2S / DRD2S
$11,600.00
M00477
293/D4 Dopamine D4 / DRD4
$11,600.00
Coming soon
CHO-K1/D5/Gα15 Dopamine D5 / DRD5
$11,600.00
CHO-K1/EDNRA Endothelin EDNRA
$11,600.00
CHO-K1/EDNRB Endothelin EDNRB
$11,600.00
CHO-K1/FFA1/Gα15 Free Fatty Acid FFA1 / GPR40
$11,600.00
CHO-K1/FFA2/Gα15 Free Fatty Acid FFA2 / GPR43
$11,600.00
CHO-K1/GAL1/Gα15 Galanin GAL1
$11,600.00
CHO-K1/GAL2 Galanin GAL2
$11,600.00
CHO-K1/GHSR Ghrelin GHSR
$11,600.00
CHO-K1/GNRHR/Gα15 Gonadotropin-releasing Hormone GNRHR
$11,600.00
293/H1 Histamine H1
$11,600.00
CHO-K1/H2/Gα15 Histamine H2
$11,600.00
CHO-K1/H3/Gα15 Histamine H3
$11,600.00
CHO-K1/H4/Gα15 Histamine H4
$11,600.00
CHO-K1/KiSS1 KiSS1-derived Peptide KiSS1 / GPR54
$11,600.00
CHO-K1/CysLT1/Gα15 Leukotriene CysLT1
$11,600.00
CHO-K1/CysLT2 Leukotriene CysLT2
$11,600.00
CHO-K1/LTB4/Gα15 Leukotriene LTB4
$11,600.00
M00488
CHO-K1/OXE-Flag/Gα15 Leukotriene OXE / OXER1
$11,600.00
Coming soon
M00463
RH7777/EDG4 Lysophospholipid EDG4 / LPA2
$11,600.00
Coming soon
M00465
RH7777/EDG6 Lysophospholipid EDG6 / S1P4
$11,600.00
Coming soon
293/MCH1 Melanin-concentrating Hormone MCH1
$11,600.00
CHO-K1/MCH2 Melanin-concentrating Hormone MCH2
$11,600.00
CHO-K1/MC2/Gα15 Melanocortin MC2
$11,600.00
CHO-K1/MC3/Gα15 Melanocortin MC3
$11,600.00
293/MC3/CRE-Luc Melanocortin MC3
$11,600.00
CHO-K1/MC4/Gα15 Melanocortin MC4
$11,600.00
CHO-K1/MC5/Gα15 Melanocortin MC5
$11,600.00
CHO-K1/MT1/Gα15 Melatonin MT1 / MTNR1A
$11,600.00
CHO-K1/MT2/Gα15 Melatonin MT2 / MTNR1B
$11,600.00
CHO-K1/MTLR/Gα15 Motilin MTLR
$11,600.00
CHO-K1/NMU1 Neuromedin U NMU1
$11,600.00
293T/NMU2 Neuromedin U NMU2
$11,600.00
M00452
CHO-K1/NPBW1/Gα15 Neuropeptide B/W NPBW1 / GPR7
$11,600.00
Coming soon
CHO-K1/NPFF1/Gα15 Neuropeptide FF NPFF1 / GPR147
$11,600.00
M00474
CHO-K1/NPFF2/Gα15 Neuropeptide FF NPFF2 / GPR74
$11,600.00
Coming soon
CHO-K1/NPS1a/Gα15 Neuropeptide S NPS1a
$11,600.00
CHO-K1/NPS1b/Gα15 Neuropeptide S NPS1b
$11,600.00
M00192
CHO-K1/NPY1/Gα15 Neuropeptide Y NPY1
$11,600.00
Coming soon
M00430
293/NPY1 Neuropeptide Y NPY1
$11,600.00
Coming soon
M00460
CHO-K1/NPY2/Gqi5 Neuropeptide Y NPY2
$11,600.00
Coming soon
CHO-K1/NPY4/Gα15 Neuropeptide Y NPY4 / PPYR1
$11,600.00
CHO-K1/NTS1 Neurotensin NTS1
$11,600.00
CHO-K1/NIACR1/Gα15 Nicotinic Acid NIACR1 / GPR109A
$11,600.00
CHO-K1/FPR1/Gα15 N-Formyl Peptide FPR1
$11,600.00
CHO-K1/FPRL1/Gα15 N-Formyl Peptide FPRL1
$11,600.00
CHO-K1/OPRD1/Gα15 Opioid OPRD1
$11,600.00
CHO-K1/OPRK1/Gα15 Opioid OPRK1
$11,600.00
CHO-K1/OPRL1/Gα15 Opioid OPRL1
$11,600.00
CHO-K1/OPRM1/Gα15 Opioid OPRM1
$11,600.00
CHO-K1/OX1 Orexin OX1
$11,600.00
CHO-K1/OX2 Orexin OX2
$11,600.00
CHO-K1/OXTR Oxytocin OT / OXTR
$11,600.00
CHO-K1/GPR103/Gα15 Peptide P518 GPR103
$11,600.00
CHO-K1/PTAFR Platelet Activating Factor PAF / PTAFR
$11,600.00
CHO-K1/PRLHR Prolactin Releasing Peptide PRLHR
$11,600.00
M00453
CHO-K1/DP1/Gα15 Prostanoid DP1 / PTGDR
$11,600.00
Coming soon
CHO-K1/DP2/Gα15 Prostanoid DP2 / GPR44
$11,600.00
293/FP/Gα15 Prostanoid FP / PTGFR
$11,600.00
293/EP1 Prostanoid EP1 / PTGER1
$11,600.00
CHO-K1/EP2/Gα15 Prostanoid EP2 / PTGER2
$11,600.00
M00485
293/EP4 Prostanoid EP4 / PTGER4
$11,600.00
Coming soon
CHO-K1/IP1/Gα15 Prostanoid IP1 / PTGIR
$11,600.00
293/TP Prostanoid TP / TBXA2R
$11,600.00
CHO-K1/PAR2/Gα15 Proteinase-activated Receptor PAR2 / F2RL1
$11,600.00
CHO-K1/PAR4 Proteinase-activated Receptor PAR4 / F2RL3
$11,600.00
CHO-K1/GPR68/Gα15 Proton-sensor GPR68
$11,600.00
1321N1/P2Y1 Purinergic P2Y1
$11,600.00
1321N1/P2Y2 Purinergic P2Y2
$11,600.00
1321N1/P2Y4 Purinergic P2Y4
$11,600.00
1321N1/P2Y6 Purinergic P2Y6
$11,600.00
1321N1/P2Y11 Purinergic P2Y11
$11,600.00
1321N1/P2Y12 Purinergic P2Y12
$11,600.00
CHO-K1/5-HT1A/Gα15 Serotonin 5-HT1A / HTR1A
$11,600.00
CHO-K1/5-HT2A Serotonin 5-HT2A / HTR2A
$11,600.00
CHO-K1/5-HT2B Serotonin 5-HT2B / HTR2B
$11,600.00
CHO-K1/5-HT2C Serotonin 5-HT2C / HTR2C
$11,600.00
HEK293/5-HT2C Serotonin 5-HT2C / HTR2C
$11,600.00
CHO-K1/5-HT4/Gα15 Serotonin 5-HT4 / HTR4
$11,600.00
293/5-HT7/CRE-Luc Serotonin 5-HT7 / HTR7
$11,600.00
CHO-K1/SST2/Gα15 Somatostatin SST2
$11,600.00
CHO-K1/SST3/Gα15 Somatostatin SST3
$11,600.00
CHO-K1/SST4/Gα15 Somatostatin SST4
$11,600.00
CHO-K1/SST5/Gα15 Somatostatin SST5
$11,600.00
CHO-K1/NK1 Tachykinin NK1 / TACR1
$11,600.00
CHO-K1/NK2 Tachykinin NK2 / TACR2
$11,600.00
CHO-K1/NK3 Tachykinin NK3 / TACR3
$11,600.00
CHO-K1/TRH1 Thyrtropin-releasing Hormone TRH1
$11,600.00
CHO-K1/UT2/Gα15 Urotensin UT2
$11,600.00
CHO-K1/V1A Vasopressin V1A / AVPR1A
$11,600.00
CHO-K1/V1B Vasopressin V1B / AVPR1B
$11,600.00
CHO-K1/V2/Gα15 Vasopressin V2 / AVPR2
$11,600.00
CHO-K1/GPR120/Gα15 Orphan GPR120
$11,600.00
M00467
CHO-K1/MRGPRD/Gα15 Orphan MRGD / MRGPRD
$11,600.00
Coming soon
CHO-K1/MRGPRX2 Orphan MRGX2 / MRGPRX2
$11,600.00
M00482
CHO-K1/OXGR1/Gα15 Orphan OXGR1
$11,600.00
Coming soon
M00472
RH7777/P2Y5 Orphan P2Y5
$11,600.00
Coming soon
M00471
CHO-K1/SUCNR1/Gα15 Orphan SUCNR1 / GPR91
$11,600.00
Coming soon
CHO-K1/CT/Gα15 Calcitonin CALCR / CT
$11,600.00
M00350
CHO-K1/AMY1/CRE-Luc Calcitonin AMY1 (RAMP1 + CALCR)
$11,600.00
Coming soon
M00478
CHO-K1/AMY2/Gα15 Calcitonin AMY2 (RAMP2 + CALCR)
$11,600.00
Coming soon
M00450
CHO-K1/AM1 Calcitonin AM1 (RAMP2 + CALCRL)
$11,600.00
Coming soon
M00479
CHO-K1/AM2/Gα15 Calcitonin AM2 (RAMP3 + CALCRL)
$11,600.00
Coming soon
CHO-K1/CRF1/Gα15 Corticotropin Releasing Factor CRF1
$11,600.00
CHO-K1/CRF2/Gα15 Corticotropin Releasing Factor CRF2
$11,600.00
CHO-K1/GCGR/Gα15 Glucagon GCGR
$11,600.00
HEK293/GCGR/Gα15 Glucagon GCGR
$11,600.00
293/GHRH/Gα15 Glucagon GHRH
$11,600.00
M00486
CHO-K1/GIP/Gα15 Glucagon GIP
$11,600.00
Coming soon
CHO-K1/GLP1/Gα15 Glucagon GLP1
$11,600.00
CHO-K1/GLP2/Gα15 Glucagon GLP2
$11,600.00
CHO-K1/SCTR/Gα15 Glucagon SCTR
$11,600.00
CHO-K1/PTH1/Gα15 Parathyroid Hormone PTH1
$11,600.00
293/PTH2/CRE-Luc Parathyroid Hormone PTH2
$11,600.00
CHO-K1/PAC1/Gα15 VIP / PACAP PAC1
$11,600.00
CHO-K1/VPAC1/Gα15 VIP / PACAP VPAC1
$11,600.00
CHO-K1/VPAC2/Gα15 VIP / PACAP VPAC2
$11,600.00
CHO-K1/CASR Calcium-sensor CASR
$11,600.00
CHO-K1/GRM2/Gα15 Glutamate mGlu2 / GRM2
$11,600.00
CHO-K1/CRE-Luc Control  
$11,600.00
293/CRE-Luc Control  
$11,600.00
CHO-K1/Gα15 Control  
$11,600.00
CHO-K1/Gqi5 Control  
$11,600.00

All the GPCRs are available as Ready-to-UseTM frozen cells.
A part of the GPCRs are available as Membrane Preparations.

Ion Channel Stable Cell Lines

Name
Type
Channel
Accession Number
CHO-K1/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/hKv1.5 Potassium, voltage-gated hKv1.5
NM_002234
HEK293/hKv4.2 Potassium, voltage-gated hKv4.2
NM_012281
HEK293/hNav1.5 Sodium, voltage-gated hNav1.5
NM_000335
HEK293/hNav1.7 Sodium, voltage-gated hNav1.7
NM_002977

Email: bioassay@genscript.com
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